Falling asleep is a complex physiological process that involves a series of stages and the interaction of multiple neurotransmitters, hormones, and neural networks. This intricate interplay ensures a smooth transition from wakefulness to sleep, allowing your body and mind to rest and rejuvenate effectively. Experience deeper, more restful sleep with our potent blend of natural ingredients.
Gamma-aminobutyric acid (GABA): GABA is the brain's primary inhibitory neurotransmitter for promoting relaxation and sleep. GABA binds to specific receptors on neurons, opening ion channels that allow negatively charged ions to enter, thereby reducing neuronal activity. This action counteracts excitatory neurotransmitters like glutamate, helping maintain the balance necessary for a healthy sleep-wake cycle. The calming effect achieved by decreased neural activity aids in transitioning from lighter stages of sleep to deeper, more restorative stages.
Although it is thought that GABA cannot pass the blood-brain barrier, it can influence the vagal afferent signals, which affect central nervous system (CNS) functions, including mood, stress response, and cognitive processes. The vagus nerve has afferent (sensory) and efferent (motor) fibres, with about 80% being afferent. These fibres convey sensory information from the gut to the brain, influencing brain function and behaviour.
Vagus Nerve: The vagus nerve is a crucial component of the gut-brain axis, facilitating rapid communication between the gut and the brain. GABA can influence vagal afferent signals, affecting CNS functions such as mood, stress response, and cognitive processes.
ENS to CNS: GABAergic neurons in the ENS communicate with the CNS through spinal and vagal pathways, contributing to regulating digestive processes and feedback to the brain.
Passion Flower Extract: Passion Flower Extract aids deep sleep by interacting with GABA receptors in the central nervous system. Reducing anxiety and inducing a state of calm can help prepare the body for sleep. Some compounds in passion flowers, such as flavonoids and alkaloids, have been shown to have mild sedative effects. This can help not only in falling asleep but also in achieving deeper, more restorative stages of sleep. The antispasmodic properties of passion flowers may help relax tense muscles, further facilitating sleep onset. This could be particularly helpful for those whose sleep is disrupted due to physical discomfort or restlessness.
Ziziphus Spinosa: Also known as jujube seed, Ziziphus Spinosa helps you fall asleep faster by naturally calming the mind and body. Rich in saponins and flavonoids, Ziziphus Spinosa increases levels of GABA in the brain, reducing neural activity and promoting relaxation. It also supports serotonin regulation, enhancing mood and aiding sleep onset. This powerful herb helps you fall asleep quickly and improves sleep quality, ensuring you wake up refreshed and rejuvenated.
Magnesium Citrate: Magnesium acts as a cofactor for activating GABA receptors. GABA inhibits neural activity, promoting relaxation and sleep. By supporting GABA function, magnesium further enhances its calming effects, making it easier to achieve a restful night's sleep. Magnesium is also involved in converting tryptophan to serotonin. This neurotransmitter subsequently converts to melatonin, a hormone that regulates sleep-wake cycles.
Furthermore, Magnesium Citrate helps with muscle function by promoting relaxation, preventing cramps and spasms, and aiding in energy production. It balances calcium levels to prevent excessive contraction, supports ATP production for energy, and helps remove lactic acid to reduce soreness. Additionally, it maintains electrolyte balance and supports protein synthesis for muscle repair and growth. These effects make magnesium citrate beneficial for overall muscle health and function.
Valerian Root: Valerian root helps you fall asleep faster by increasing levels of GABA in the brain. This promotes relaxation and reduces anxiety. Valerian root works by inhibiting the breakdown of GABA, enhancing its calming effects on the nervous system. Additionally, the valerian root contains:
- Compounds with sedative properties.
- Soothing both mind and body.
- Supporting a quicker transition to sleep and improving sleep quality.
Corydalis Yanhusuo: Corydalis Yanhusuo is a traditional herbal remedy widely used in Traditional Chinese Medicine. It helps you fall asleep faster by acting as a natural sedative and pain reliever. It increases levels of GABA in the brain, calming the nervous system and reducing anxiety. Additionally, Corydalis Yanhusuo contains compounds that inhibit dopamine receptors, helping to alleviate pain and promote relaxation. This dual action eases discomfort and induces a tranquil state, making it easier to drift into a restful sleep.
L-Theanine: L-Theanine helps you fall asleep faster by promoting relaxation and reducing stress without causing drowsiness. This amino acid, commonly found in green tea, increases calming neurotransmitters such as GABA, serotonin, and dopamine levels in the brain. These neurotransmitters calm the mind and reduce anxiety, making it easier to drift into sleep. Additionally, L-Theanine enhances alpha brain waves, which are associated with a relaxed yet alert state, further facilitating a smooth transition to sleep.
L-Tyrosine: L-tyrosine, an amino acid, helps you fall asleep faster by supporting the production of neurotransmitters that regulate mood and stress levels. By promoting the synthesis of dopamine, norepinephrine, and epinephrine, L-tyrosine stabilises mood and reduces stress, creating a relaxed state conducive to sleep. Additionally, it replenishes neurotransmitters depleted by stress and fatigue, ensuring optimal brain function and a smooth transition into sleep.
5-HTP: 5-HTP is a naturally occurring amino acid derivative produced in the body from tryptophan. It indirectly boosts melatonin production by increasing serotonin levels, aiding sleep. Some studies suggest that 5-HTP can improve sleep quality by prolonging the REM phase, although further research is needed. Enhancing serotonin and melatonin levels, 5-HTP may contribute to deeper, more restorative sleep.
Zinc Sulphate: Zinc Sulphate helps you fall asleep faster by supporting the production and regulation of melatonin, the hormone responsible for sleep-wake cycles. By enhancing melatonin levels, Zinc Sulphate helps establish a consistent sleep pattern and improves sleep quality. Additionally, zinc plays a crucial role in neurotransmitter function and reduces inflammation, contributing to a more relaxed and restful state.
Vitamin B6 (Pyridoxine): Vitamin B6 helps you fall asleep faster by playing a crucial role in producing serotonin and melatonin, two essential hormones that regulate sleep. Serotonin promotes relaxation and mood stability, while melatonin controls your sleep-wake cycle. By boosting the synthesis of these hormones, Vitamin B6 calms the nervous system, making it easier to drift into sleep. Additionally, Vitamin B6 supports overall brain health and reduces symptoms of stress and anxiety, further enhancing sleep quality.